COMPETITIVE MOLECULES = SIMILAR SHAPE TO SUBSTRATE
- COMPETE WITH SUBSTRATE FOR ACTIVE SITE
- NO REACTION TAKES PLACE
BLOCK ACTIVE SITE
- NO SUBSTRATE CAN BIND
HIGH CONC OF INHIBITOR
- MORE ACTIVE SITES OCCUPIED
- FEW E.S.C
HIGHER CONC OF SUBSTRATE
- INCREASE R.O.R
- GET TO ACTIVE SITE QUICKER
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